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  • Endothelin Receptor Antagonist
    3 Drugs classified under this drug class


    All the Drug Class Drugs

    Opsumit
    Actelion
    RX
    partial basket chart
    Opsumit

    Endothelin Receptor Antagonist. Macitentan 10 mg.
    F.C. TABS.: 30. 10 mg ×1/d, with or
    without food, should be taken every
    day at the same time.
    Tmt. of PAH, who GROUP I to delay dis.
    progress. Dis. progress. includ. : death,
    initiat. of IV or subcutan. prostanoids, or
    clin. worsening of PAH (decreased 6-min.
    walk distance, worsened PAH sympt. and
    need for additional PAH tmt.). The drug
    also reduced hospitaliz. for PAH.
    C/I: Hypersens., Preg., WOCBP who are
    not using reliable contracep., Lact. Pts.
    with severe hep. impair. (with or without
    cirrhosis). Baseline values of hep.
    aminotransferases (AST and/or ALT > 3 ×
    ULN).

    Tracleer
    Actelion
    RX
    partial basket chart
    Tracleer

    Endothelin Receptor Antagonist. Bosentan 62.5 mg, 125 mg.
    F.C. TABS: 60 x 62.5 mg, 125 mg. Initial:
    62.5 mg 2 x dly for 4 wks. Maint: 125 mg
    2 x dly morn. and even. with or without
    food.
    Prim. pulm. arterial hypertens. or second.
    to scleroderma or other connect. tissue
    dis. Reduct. number new digital ulcs. in
    system. sclerosis, ongoing digital ulc. dis.
    C/I: Pregn.

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